Permeability | Permeability | |
Caco-2 cells permeability |
|
MDCK cells permeability |
|
PAMPA membrne Permeability |
Plasma protein binding | Plasma protein binding | |
Plasma protein binding assay |
Drug metabollism | Metabolic stabililty | |
Plasma stability |
|
Microsomal stability |
|
Hepatocyte stability |
Metabolite profiling & ID | |
Metabolite profiling & ID |
Drug metabollism Reaction phenotyping | |
Reaction phenotyping for CYP (recombinant CYPs) |
|
Reaction phenotyping for UGT (recombinant UGTs) |
Drug transporter | Drug transporter Reaction phenotyping | |
Reaction phenotyping for Transport |
|
Reaction phenotyping for Transport (Kinetic study) |
Drug-Drug interaction | Enzyme Inhibition | |
CYP Inhibition (Screening of CYP inhibition) |
|
CYP inhibition (IC50 assay) |
|
CYP inhibition (Ki assay) |
|
UGT Inhibition (Screening of UGT inhibition) |
|
UGT Inhibition (IC50 assay) |
|
UGT inhibition (Ki assay) |
|
Time-Dependent Inhibition (IC50 shift assay) |
|
Time-Dependent Inhibition (Kinact/KI assay) |
|
Microsomal binding assay |
Transporter Inhibition | |
Transporter Inhibition (Screening) |
|
Transporter Inhibition (IC50 assay) |
|
Transporter Inhibition (Ki assay) |
|
Transporter inhibition (Time-Dependent Inhibition, IC50 shift assay) |
Enzyme/Transporter Induction | |
Enzyme/Transporter Induction |
|
Enzyme Induction (EC50 assay) |
|
PXR reporter assay |
|
Cell viability |
Bioanalytical services | Bioanalytical service | |
약물분석법개발 |
|
In vivo PK 혈장 분석 |
Preclinical study |
- |
|
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